Page last updated: 2024-08-21

2,4-pyridinedicarboxylic acid and 3-[[2-(2-pyridinyl)-6-(1,2,4,5-tetrahydro-3-benzazepin-3-yl)-4-pyrimidinyl]amino]propanoic acid

2,4-pyridinedicarboxylic acid has been researched along with 3-[[2-(2-pyridinyl)-6-(1,2,4,5-tetrahydro-3-benzazepin-3-yl)-4-pyrimidinyl]amino]propanoic acid in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's3 (75.00)24.3611
2020's1 (25.00)2.80

Authors

AuthorsStudies
Brennan, PE; Burgess-Brown, NA; Che, K; Daniel, M; England, KS; Kawamura, A; Krojer, T; Ng, SS; Schofield, CJ; Scozzafava, G; Szykowska, A; Tumber, A; von Delft, F1
Athanasou, N; Badock, V; Brennan, PE; Brown, J; Burgess-Brown, N; Egner, U; Gileadi, C; Hookway, ES; Johansson, C; Kopec, J; LaThangue, NB; Munro, S; Nowak, RP; Nuzzi, A; Oppermann, U; Philpott, M; Prinjha, R; Steuber, H; Strain-Damerell, C; Szykowska, A; Tumber, A; Velupillai, S; Westaway, S; Wu, N1
Abboud, MI; Langley, GW; Lohans, CT; Schofield, CJ1
Andrijes, R; Ansari, MSZ; Antonini, L; Ciogli, A; Coleman, ML; Del Bufalo, D; Hendrix, E; Johansson, C; Kawamura, A; Mai, A; Mautone, N; Nowak, RP; Oppermann, U; Passeri, D; Pellegrini, FR; Pellicciari, R; Ragno, R; Rotili, D; Sabatino, M; Salah, E; Schofield, CJ; Simelis, K; Trisciuoglio, D; Tumber, A1

Other Studies

4 other study(ies) available for 2,4-pyridinedicarboxylic acid and 3-[[2-(2-pyridinyl)-6-(1,2,4,5-tetrahydro-3-benzazepin-3-yl)-4-pyrimidinyl]amino]propanoic acid

ArticleYear
Optimisation of a triazolopyridine based histone demethylase inhibitor yields a potent and selective KDM2A (FBXL11) inhibitor.
    MedChemComm, 2014, Dec-01, Volume: 5, Issue:12

    Topics:

2014
Structural analysis of human KDM5B guides histone demethylase inhibitor development.
    Nature chemical biology, 2016, Volume: 12, Issue:7

    Topics: Antineoplastic Agents; Cell Proliferation; Drug Screening Assays, Antitumor; Enzyme Inhibitors; Histone Demethylases; Humans; Jumonji Domain-Containing Histone Demethylases; Models, Molecular; Multiple Myeloma; Nuclear Proteins; Protein Conformation; Repressor Proteins; Structure-Activity Relationship

2016
Inhibition of a viral prolyl hydroxylase.
    Bioorganic & medicinal chemistry, 2019, 06-15, Volume: 27, Issue:12

    Topics: Enzyme Assays; Hydroxylation; Hypoxia-Inducible Factor-Proline Dioxygenases; Ketoglutaric Acids; Oligopeptides; Phycodnaviridae; Procollagen-Proline Dioxygenase; Prolyl-Hydroxylase Inhibitors; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization

2019
First-in-Class Inhibitors of the Ribosomal Oxygenase MINA53.
    Journal of medicinal chemistry, 2021, 12-09, Volume: 64, Issue:23

    Topics: Cell Line, Tumor; Cell Proliferation; Crystallization; Dioxygenases; Enzyme Inhibitors; Histone Demethylases; Humans; Models, Molecular; Nuclear Proteins; Protein Conformation; Ribosomes; Substrate Specificity

2021